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| Product Name | TC-G 1008 |
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| Description | Potent and selective GPR39 agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively). Selective over a panel of kinases (IC50s > 10 μM) and displays minimal binding affinity for ghrelin and neurotensin-1 receptors (IC50s > 30 μM). Increases GLP-1 levels in vitro and in vivo. Orally bioavailable. Purity 98%. MW (observed): 418.9 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide |
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| Gene, Accession, CAS # | CAS: 1621175-65-2 |
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| Catalog # | 5355/10 |
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| Price | |
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| Order / More Info | TC-G 1008 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 27235821, 30419533, 30459126 |
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| 产品资料 |
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