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| Product Name | EPZ 015666 |
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| Description | Potent and selective protein arginine methyltransferase 5 (PRMT5) inhibitor (IC50 = 22 nM, Ki = 5 nM). Displays selectivity for PRMT5 over a panel of 20 other protein methyltransferases. Exhibits dose-dependent antitumor effects in multiple mantle cell lymphoma (MCL) xenograft models. Orally bioavailable. Purity 98%. MW (observed): 383.44 |
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| Size | 25 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-[(2S)-3-(3,4-Dihydro-2(1H)-isoquinolinyl)-2-hydroxypropyl]-6-(3-oxetanylamino)-4-pyrimidinecarboxamide |
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| Gene, Accession, CAS # | CAS: 1616391-65-1 |
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| Catalog # | 6516/25 |
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| Price | |
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| Order / More Info | EPZ 015666 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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