产品名称 AZ 3451 from TOCRIS BIOSCIENCE
产品货号 6806/10
产品价格 现货询价,电话:010-67529703
产品规格 10 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameAZ 3451
DescriptionPotent allosteric PAR2 antagonist (IC50 = 23 nM); binds to a remote allosteric site outside the helical bundle. Inhibits ERK phosphorylation in 1321N1 cells overexpressing wild-type human PAR2. Highly lipophilic. Purity 98%. MW (observed): 571.46
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names2-(6-Bromo-1,3-benzodioxol-5-yl)-N-(4-cyanophenyl)-1-[(1S)-1-cyclohexylethyl]-1H-benzimidazole-5-carboxamide
Gene, Accession, CAS #CAS: 2100284-59-9
Catalog #6806/10
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Order / More InfoAZ 3451 from TOCRIS BIOSCIENCE
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