产品名称 NVP DPP 728 dihydrochloride from TOCRIS BIOSCIENCE
产品货号 3506/50
产品价格 现货询价,电话:010-67529703
产品规格 50 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameNVP DPP 728 dihydrochloride
DescriptionPotent, orally active dipeptidyl peptidase (DPP)-IV inhibitor (Ki = 11 nM, IC50 = 14 nM) that displays > 15 000-fold selectivity over DPP-II and a range of proline-cleaving proteases. Exhibits antidiabetic activity in vivo; improves glucose tolerance, increases glucagon-like peptide 1 (GLP-1) and insulin levels, augments insulin secretion and GLUT2 levels, and reduces (preserves) islet size. Purity 97%. MW (observed): 371.27
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names6-[[2-[[2-(2S)-2-Cyano-1-pyrrolidinyl]-2-oxoethyl]amino]ethyl]amino-3-pyridinecarbononitrile dihydrochloride
Gene, Accession, CAS #CAS: 207556-62-5
Catalog #3506/50
Price
Order / More InfoNVP DPP 728 dihydrochloride from TOCRIS BIOSCIENCE
Product Specific ReferencesPubMed: 22821947
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