| 产品详情 |
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| Product Name | GSK 1702934A |
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| Description | Potent and selective TRPC3/6 activator (EC50 = 80 and 440 nM for TRPC3 and 6, respectively). Exhibits no activity at TRPV4, TRPA1, M1, M4, CaV1.2, hERG, NaV1.5, or CXCR5 receptors at concentrations <10 μmol/L. Induces TRPC3/6-currents in HEK293 cells transduced with recombinant human TRPC3/6. Directly activates TRPC channels through by-passing phospholipase-C signaling. Also induces calcium signals in HEK-TRPC6 cells (pEC50 = 6.6). Purity 98%. MW (observed): 395.52 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 1,3-Dihydro-1-[1-[(5,6,7,8-tetrahydro-4H-cyclohepta[b]thien-2-yl)carbonyl]-4-piperidinyl]-2H-benzimidazol-2-one |
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| Gene, Accession, CAS # | CAS: 924377-85-5 |
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| Catalog # | 6508/50 |
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| Price | |
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| Order / More Info | GSK 1702934A from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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| 产品资料 |
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