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| Product Name | J 104129 fumarate |
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| Description | Potent M3 muscarinic receptor antagonist that displays ~ 120-fold selectivity over M2 receptors (Ki values are 4.2, 19 and 490 nM for human M3, M1 and M2 receptors respectively). Exhibits > 250-fold bronchial selectivity; inhibits ACh-induced bronchoconstriction but not ACh-induced bradycardia (KB values are 3.3 and 170 nM for rat trachea M3 and rat right atria M2 receptors respectively). Purity 99%. MW (observed): 500.63 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-pentenyl)-4-piperidinyl]benzeneacetamide fumarate |
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| Gene, Accession, CAS # | CAS: 257603-40-0 |
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| Catalog # | 2507/10 |
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| Order / More Info | J 104129 fumarate from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 26236483 |
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