产品名称 PI 3065 from TOCRIS BIOSCIENCE
产品货号 5919/50
产品价格 现货询价,电话:010-67529703
产品规格 50 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NamePI 3065
DescriptionPotent and selective PI 3-kinase p110δ inhibitor (IC50 = 5 nM; Ki = 1.5 nM). Exhibits >100-fold selectivity over p100α, p100γ and p100β isoforms (IC50 values are 600, 910, >10,000 nM, respectively). Attenuates 4TI tumor growth and metastasis in vivo. Purity 98%. MW (observed): 506.64
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names6-[[4-(Cyclopropylmethyl)-1-piperazinyl]methyl]-2-(5-fluoro-1H-indol-4-yl)-4-(4-morpholinyl)-thieno[3,2-d]pyrimidine
Gene, Accession, CAS #CAS: 955977-50-1
Catalog #5919/50
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Order / More InfoPI 3065 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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