| 产品详情 |
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| Product Name | GSK343 |
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| Description | A potent histone H3-lysine 27 (H3K27) methyltransferase EZH2 inhibitor (IC50 = 4 nM). Diplays 1000-fold selectivity for other HMTs except EZH1 (60-fold selectivity). GSK343 inhibits H3K27 methylation in HCC1806 cells with an IC50 of <200nM (measured by immunofluorescence). MW: 541.69. Purity ≥99% by HPLC |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 1-Isopropyl-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-6-(2-(4-methylpiperazin-1-yl)pyridine-4-yl)-1H-indazole-4-carboxamide |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 2281-5 |
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| Price | |
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| Order / More Info | GSK343 from BIOVISION, INC. |
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| Product Specific References | n/a |
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