| 产品详情 |
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| Product Name | GSK-2126458 |
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| Description | MW: 505.5. Purity ≥98% by HPLC. Background: Cell-permeable. A highly potent, pan phosphoinositide 3-kinase (PI 3-K) family kinase inhibitor with biochemical Ki's of 0.019 nM (PI 3-K?), 0.13 nM (PI 3-Kbeta), 0.024 nM (PI 3-Kdelta), 0.06 nM (PI 3-K?), 0.18 nM (mTORC1), and 0.3 nM (mTORC2). In vivo, GSK2126458 displays anti-tumor activity in both pharmacodynamic and tumor growth efficacy models. |
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| Size | 1 mg, 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | [2,4-Difluoro-N-{2-(methyloxy)-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl}benzenesulfonamide] |
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| Gene, Accession, CAS # | CAS: 1086062-66-9 |
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| Catalog # | MBS842084 |
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| Order / More Info | GSK-2126458 from MYBIOSOURCE INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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