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| Product Name | GF 109203X |
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| Description | Very potent and selective inhibitor of protein kinase C, selective for the α and β1 isoforms (IC50 values are 0.0084, 0.0180, 0.210, 0.132, and 5.8 μM for α, β1, δ, ε and ζ isoforms respectively). Selective over MLCK, PKG and PKA (IC50 values are 0.6, 4.6, and 33 μM respectively). Potent antagonist at the 5-HT3 receptor (Ki = 29.5 nM). Anti-inflammatory in vivo. Purity 98%. MW (observed): 412.49 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 2-[1-(3-Dimethylaminopropyl)indol-3-yl]-3-(indol-3-yl) maleimide. Gö 6850, Bisindolylmaleimide I |
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| Gene, Accession, CAS # | CAS: 133052-90-1 |
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| Catalog # | 0741/10 |
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| Order / More Info | GF 109203X from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 11087819, 12642376, 12880426, 15901799, 16672661, 17277031, 17592023, 17923483, 18094230, 18724384, 19298234, 19846725, 21068362, 21593487, 21653882, 21949111, 21957263, 22155728, 22220695, 22275752, 22492526, 23269840, 23400781, 24078773, 24258815, 24335212, 24908484, 24916153, 25261977, 25617350, 25768340, 26019328, 26241492, 26245668, 26510981, 26655905, 26667040, 26909238, 27396242, 29966616 |
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