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| Product Name | UNC 0646 |
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| Description | Potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50 values are 6 nM and 15 nM for G9a and GLP, respectively). Potently blocks G9a/GLP methyltransferase activity in cells (IC50 = 10 nM in MCF7 cells); exhibits low cellular toxicity (EC50 = 4.7 μM in MCF7 cells). Selective for G9a/GLP over a range of other protein lysine methyltransferases and protein arginine methyltransferases. Purity 99%. MW (observed): 621.9 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-(1-Cyclohexyl-4-piperidinyl)-2-[hexahydro-4-(1-methylethyl)-1H-1,4-diazepin-1-yl]-6-methoxy-7-[3-(1-piperidinyl)propoxy]-4-quinazolinamine |
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| Gene, Accession, CAS # | CAS: 1320288-17-2 |
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| Catalog # | 4342/10 |
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| Price | |
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| Order / More Info | UNC 0646 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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| 产品资料 |
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