| 产品详情 |
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| Product Name | Octreotide (acetate) |
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| Description | A somatostatin receptor agonist (Kis = 875, 0.57, 26.8, >1,000, and 6.8 nM for SST1-5 receptors, respectively); selectively binds to SST2 over SST3 and SST5 receptors (IC50s = 0.02, 92.9, and 21.8 nM, respectively); inhibits the secretion of growth hormone in vitro in rat pituitary cells three-fold more potently than somatostatin; inhibits the secretion of growth hormone in vivo in rhesus monkey (ID50 = 0.38 µg/kg per hour); inhibits proliferation of VEGF-stimulated human umbilical endothelial cells (HUVECs) with an EC50 value of approximately 1 µM; inhibits growth of LCI-D20 human hepatocellular carcinoma cell tumors in a nude mouse xenograft model when administered at a dose of 50 µg/kg twice daily |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | SMS 201-995 |
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| Gene, Accession, CAS # | CAS: 760176-26-9 |
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| Catalog # | 23757-10 |
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| Order / More Info | Octreotide (acetate) from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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