| 产品详情 |
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| Product Name | Netupitant |
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| Description | An NK1 receptor antagonist (Ki = 0.95 nM); selective for human NK1 over human NK2 and NK3 and rat NK1 (Kis = >1,500 nM); selective for NK1 over 50 G protein-coupled receptors, monoamine transporters, and ion channels when used in the nanomolar range; decreases the maximal response to substance P in isolated guinea pig ileum; inhibits substance P-induced scratching, biting, and licking in mice at doses of 1-10 mg/kg; decreases NK agonist-induced foot tapping in gerbils (ID50s = 1.5 mg/kg, i.p., or 0.5 mg/kg, oral). |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | Ro 67-31898/000 |
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| Gene, Accession, CAS # | CAS: 290297-26-6 |
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| Catalog # | 23809-50 |
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| Price | |
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| Order / More Info | Netupitant from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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