产品名称 L Moses dihydrochloride from TOCRIS BIOSCIENCE
产品货号 6251/10
产品价格 现货询价,电话:010-67529703
产品规格 10 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameL Moses dihydrochloride
DescriptionHigh affinity and selective cell-permeable p300/CBP-associated factor (PCAF) inhibitor (Ki = 47 nM). Exhibits no significant activity against a panel of 48 other bromodomains except GCN5 (Kd = 600 nM). Exhibits >4500-fold selectivity for PCAF over BRD4. Also exhibits metabolic stability in mouse and human liver microsomes and no observable cytotoxicity in peripheral blood mononuclear cells (PBMC). Purity 98%. MW (observed): 433.38
Size10 mg
Concentrationn/a
Applicationsn/a
Other Names(1S, 2S)-N1,N1-Dimethyl-N2-(3-methyl-1,2,4-triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diamine dihydrochloride
Gene, Accession, CAS #n/a
Catalog #6251/10
Price
Order / More InfoL Moses dihydrochloride from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
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