| 产品详情 |
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| Product Name | Fendiline (hydrochloride) |
| Description | An α2-adrenergic receptor antagonist (Kd = 2.6 µM) and an L-type calcium channel blocker (IC50 = 17 µM) well-known for its coronary vasodilator effects; inhibits K-Ras plasma membrane localization (IC50 = 9.64 µM), blocking the proliferation of K-Ras-transformed tumor cells |
| Size | 5 g |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 119959-32-9 13042-18-7 calcium channel blocker Ca2+ antagonist vasodilation hypertension cardiology signal transduction cancer ion pump biochemical receptor vascular disease Cordan Fendilar Phenoxan Sensit Sensite α2-adrenergic L-type coronary vasodilator inhibit inhibition K-Ras KRas plasma membrane localization tumor |
| Gene, Accession, CAS # | CAS: 13636-18-5 |
| Catalog # | 17295-5 |
| Price | |
| Order / More Info | Fendiline (hydrochloride) from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
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