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| Product Name | Elagolix (sodium salt) |
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| Description | An antagonist of GnRHR (Ki = 0.9 nM in a radioligand binding assay); selective for GnRHR over CYP3A4 (IC50 = 56 µM) as well as a panel of 100 receptors, ion channels, enzymes, and transporters (IC50s = >10 µM); inhibits GnRH-induced inositol phosphate production in RBL-1 cells expressing human GnRHR (IC50 = 1.5 nM); suppresses production of luteinizing hormone in castrated male cynomolgus macaques at 30 mg/kg |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | n/a |
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| Gene, Accession, CAS # | CAS: 832720-36-2 |
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| Catalog # | 26534-10 |
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| Price | |
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| Order / More Info | Elagolix (sodium salt) from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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