产品名称 3,5-Diiodothyropropionic Acid from CAYMAN CHEMICAL COMPANY
产品货号 23299-25
产品价格 现货询价,电话:010-67529703
产品规格 25 mg
产品品牌 CAYMAN CHEMICAL COMPANY
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Product Name3,5-Diiodothyropropionic Acid
DescriptionAn inotropic thyroid hormone analogue of L-thyroxine; binds to TRα and TRβ (Kas = 2.4 and 4.06 x 107 M-1, respectively, for human recombinant receptors); increases mRNA expression of α-MHC in primary rat cardiomyocytes (EC50 = ~0.5 µM); prevents myocardial infarction-induced loss of contractility ex vivo in rabbit cardiomyocytes (3.75 mg/kg per day); increases expression of VEGF, bFGF, angiopoietin-1, and Tie-2 as well as angiogenesis in non-infarcted cardiac tissue in rats (3.75 mg/kg per day); decreases infarct size expansion, stimulates arteriolar growth, and inhibits ventricular remodeling post-myocardial infarction in rats (3.5 mg/kg per day)
Size25 mg
Concentrationn/a
Applicationsn/a
Other NamesDITPA
Gene, Accession, CAS #CAS: 1158-10-7
Catalog #23299-25
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Order / More Info3,5-Diiodothyropropionic Acid from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
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