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| Product Name | Alvimopan |
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| Description | A μ-opioid receptor antagonist (Ki = 0.47 nM); selective over κ- and δ-opioid receptors (Kis= 100 nM and 12 nM, respectively); inhibits μ-opioid receptor mediated GTP binding to CHO cell membranes (IC50 = 1.7 nM); inhibits morphine-induced slowing of colorectal transit in mice (ED50 = 0.41 mg/kg, p.o.); antagonizes morphine-but not apraclonidine-induced inhibition of GI transit in rats (0.3 and 1 mg/kg, p.o.) |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | ADL 8-2698|LY246736 |
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| Gene, Accession, CAS # | CAS: 156053-89-3 |
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| Catalog # | 23902-10 |
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| Price | |
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| Order / More Info | Alvimopan from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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