| 产品详情 |
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| Product Name | DPDPE (trifluoroacetate salt) |
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| Description | A synthetic pepetide δ-opioid receptor agonist (Ki = 2.7 nM in rat brain homogenates); >250-fold selectivity for the δ-opioid receptor over the μ- and κ-opioid receptors in rat brain homogenates (Kis = 713 and >1,500 nM, respectively); selectively inhibits electrically-evoked contractions in mouse vas deferens over guinea pig myenteric plexus (IC50s = 4.14 and 3,000 nM, respectively); completely blocks MES-induced tonic hindlimb extension in 50% of tested rats and increases the flurothyl-induced seizure threshold by 15-20% in rats at 140 nmol; reduces formalin-induced paw licking and lifting, indicating analgesia, in rats from 1-10 µg; increases the latency to tail withdrawal in the tail-immersion test in both wild-type and δ-opioid receptor knockout mice |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | [D-Pen2,D-Pen5]Enkephalin |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 23184-5 |
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| Price | |
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| Order / More Info | DPDPE (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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