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Product Name | BQ-788 Sodium Salt |
Description | BQ-788 is a potent and selective antagonist of endothelin (ET) B-receptor (IC50 = 1.2 nM). BQ-788 is a good tool for demonstrating the role of ET-1 and ET(B) receptor subtypes in physiological and/or pathophysiological conditions. Q-788 competitively antagonizes the vasoconstriction induced by an ETB-selective agonist on isolated rabbit pulmonary arteries, blocks ET-1 induced bronchoconstriction in guinea pigs, and abolishes an ET-1 mediated depressor response in rats. MW: 663.79. Purity ≥97% by HPLC |
Size | 500 µg |
Concentration | n/a |
Applications | n/a |
Other Names | (2R)-2-[[(2R)-2-amino-3-(1-methoxycarbonylindol-3-yl)propanoyl]-[(2S)-2-[[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]amino]-4,4-dimethylpentanoyl]amino]hexanoate, sodium |
Gene, Accession, CAS # | CAS: 156161-89-6 |
Catalog # | B1554-500 |
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Order / More Info | BQ-788 Sodium Salt from BIOVISION, INC. |
Product Specific References | n/a |
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