| 产品详情 |
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| Product Name | Amisulpride |
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| Description | Potent, selective dopamine D2 and D3 receptor antagonist. Ki values are 2.8 and 3.2 nM respectively for human D2 and D3 and > 1000 nM for human D1, D4 and D5 receptors. Shows selectivity for presynaptic dopamine autoreceptors at low doses and blocks postsynaptic D2/D3 receptors at higher doses. Preferentially interacts with limbic D2-like receptors in vivo. Atypical antipsychotic/antischizophrenic agent with limited extrapyrimidal side effects and a profile distinct from that of haloperidol and remoxipride. Purity 98%. MW (observed): 369.48 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 4-Amino-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-benzamide. DAN 2163 |
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| Gene, Accession, CAS # | CAS: 71675-85-9 |
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| Catalog # | 2132/50 |
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| Order / More Info | Amisulpride from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 21966518, 22817643 |
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| 产品资料 |
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