产品详情 |
Edit |   |
Product Name | BAN ORL 24 |
Description | Potent and selective NOP receptor antagonist (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). Inhibits nociceptin-induced stimulation of [35S]-GTPγS binding and Ca2+ mobilization in CHO cells in vitro and antagonizes NOP agonist-induced reduction in locomotor activity in vivo. Brain penetrant. Purity 97%. MW (observed): 506.51 |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | (2R)-1-(Phenylmethyl)-N-[3-(spiro[isobenzofuran-1(3H),4'-piperidin]-1-yl)propyl-2-pyrrolidinecarboxamide |
Gene, Accession, CAS # | CAS: 1401463-54-4 |
Catalog # | 3661/10 |
Price | |
Order / More Info | BAN ORL 24 from TOCRIS BIOSCIENCE
|
Product Specific References | PubMed: 24428821 |
产品资料 |
|
|