| 产品详情 |
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| Product Name | CRT 0066101 |
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| Description | Potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively). Exhibits selectivity for PKD against a panel of >90 protein kinases, including PKCα, MEK, ERK, c-Raf and c-Src. Reduces proliferation and cell viability of pancreatic cancer cells expressing moderate levels of endogenous PKD1/2. Orally bioavailable. Purity 98%. MW (observed): 411.33 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 2-[4-[[(2R)-2-aminobutyl]amino]-2-pyrimidinyl]-4-(1-methyl-1H-pyrazol-4-yl)phenol dihydrochloride |
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| Gene, Accession, CAS # | CAS: 1883545-60-5 |
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| Catalog # | 4975/10 |
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| Price | |
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| Order / More Info | CRT 0066101 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 25698580, 27030010 |
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| 产品资料 |
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