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| Product Name | SR 49059 |
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| Description | Potent and selective non-peptide vasopressin V1A receptor antagonist; devoid of agonist activity. Displays high affinity and efficacy at both rat (Ki = 1.6 nM) and human (Ki = 1.1 - 6.3 nM) V1A receptors. Potently antagonizes arginine vasopressin-induced effects in vitro (IC50 = 3.7 nM for inhibition of human platelet aggregation) and is orally active in vivo. Purity 99%. MW (observed): 620.5 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide. Relcovaptan |
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| Gene, Accession, CAS # | CAS: 150375-75-0 |
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| Catalog # | 2310/10 |
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| Price | |
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| Order / More Info | SR 49059 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 21256175, 21725754, 23690069, 24517977 |
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| 产品资料 |
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