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Product Name | SR 141716A |
Description | Potent and selective cannabinoid CB1 receptor antagonist (Ki = 1.98 nM). Also acts as an inverse agonist reversing adenylyl cyclase inhibition by WIN 55,212-2 (Cat.No. 1038) (IC50 = 48 nM). Displays no activity at CB2 receptors. Reduces food intake and body weight in orally dosed non-obese Wistar rats. Also μ-opioid receptor antagonist (Ki = 652 nm). Purity 99%. MW (observed): 500.25 |
Size | 50 mg |
Concentration | n/a |
Applications | n/a |
Other Names | N-(Piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide hydrochloride. Rimonabant hydrochloride |
Gene, Accession, CAS # | CAS: 158681-13-1 |
Catalog # | 0923/50 |
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Order / More Info | SR 141716A from TOCRIS BIOSCIENCE
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Product Specific References | PubMed: 10780977, 11454655, 15629705, 16864584, 18174385, 21849983, 23426954, 25411367, 25740522, 26740814, 27065006, 27404492, 27861729, 9690851 |
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