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| Product Name | EMPA |
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| Description | Highly potent, selective OX2 receptor antagonist (IC50 values are 2.3 nM and 1900 nM for OX2 and OX1 respectively). Displays negligible or no inhibition of a panel of 80 receptors. Blocks orexin-B- and orexin-A-invoked calcium mobilization in hOX2-expressing CHO cells (IC50 values are 7.9 nM and 8.8 nM respectively); reverses orexin-B-induced hyperlocomotion in mice. Brain penetrant. Purity 98%. MW (observed): 454.54 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-Ethyl-2-[(6-methoxy-3-pyridinyl)[(2-methylphenyl)sulfonyl]amino]-N-(3-pyridinylmethyl)-acetamide |
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| Gene, Accession, CAS # | CAS: 680590-49-2 |
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| Catalog # | 4558/10 |
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| Price | |
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| Order / More Info | EMPA from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 25552485, 26174505 |
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| 产品资料 |
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