| 产品详情 |
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| Product Name | Endomorphin 2 (trifluoroacetate salt) |
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| Description | An endogenous neuropeptide and μ-opioid receptor agonist (Ki = 0.69 nM); selective for μ- over δ- and κ-opioid receptors (Kis = 9,233 and 5,240 nM, respectively); binds to mouse brain membranes and rat recombinant μ-opioid receptors expressed in CHO cells (Kis = 1.37 and 0.58 nM, respectively); inhibits forskolin-induced cAMP accumulation in CHO cells expressing rat recombinant μ-opioid receptors and in SH-SY5Y human neuroblastoma cells (IC50s = 7.08 and 7.76 nM, respectively); increases analgesia in a radiant heat tail-flick assay in mice following intracerebroventricular or intrathecal administration (ED50s = 1.99 and 3.81 µg, respectively); induces conditioned place aversion in mice at 10 µg, i.c.v.; decreases gastrointestinal transit time in mice at 3 µg, i.c.v., |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | Tyr-Pro-Phe-Phe-NH2 |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 23281-5 |
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| Price | |
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| Order / More Info | Endomorphin 2 (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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