| 产品详情 |
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| Product Name | TAK 165 |
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| Description | Potent, irreversible human epithelial growth factor receptor 2 (ErbB2) inhibitor (IC50 = 6 nM) that displays > 4000-fold selectivity over EGFR, FGFR, PDGFR, JAK1 and Src. Exhibits potent antiproliferative effects in ErbB2-overexpressing cancer cell lines (IC50 = 5 nM in BT474 breast cancer cells) and significantly inhibits bladder, breast and prostate cancer xenograft growth in vivo. Purity 99%. MW (observed): 468.47 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 1-[4-[4-[[2-[(1E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-4-oxazolyl]methoxy]phenyl]butyl]-1H-1,2,3-triazole. Mubritinib |
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| Gene, Accession, CAS # | CAS: 366017-09-6 |
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| Catalog # | 3599/10 |
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| Price | |
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| Order / More Info | TAK 165 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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