产品名称 AZ 6102 from TOCRIS BIOSCIENCE
产品货号 5775/50
产品价格 现货询价,电话:010-67529703
产品规格 50 mg
产品品牌 TOCRIS BIOSCIENCE
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Product NameAZ 6102
DescriptionPotent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively). Exhibits >100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6. Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM). Exhibits moderate oral bioavailability. Purity 98%. MW (observed): 428.53
Size50 mg
Concentrationn/a
Applicationsn/a
Other Namesrel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
Gene, Accession, CAS #CAS: 1645286-75-4
Catalog #5775/50
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Order / More InfoAZ 6102 from TOCRIS BIOSCIENCE
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