| 产品详情 |
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| Product Name | Azamulin |
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| Description | MW: 478.65. Purity ≥98% by HPLC. Azamulin is a derivative of the antibiotic pleuromutilin. It is a highly selective inhibitor of the CYP3A family (IC50 = 0.03-0.24 muM as reported in Stresser et al.; DMD; January 2004 vol. 32 no. 1 p105-112). Azamulin is a 15 and 13 fold more potent inhibitor of CYP3A4 compared to CYP3A5 or CYP3A7 respectively making it very useful for CYP3A4 activity assays and can be used as a benchmark in CYP3A4 inhibitor screening assays. It is at least 100 fold selective |
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| Size | 1 mg, 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | [(5-Amino-1H-1; 2; 4-triazol-3-yl) thio]acetic acid (3aS; 4R; 5S; 6R; 8R; 9R; 9aR; 10R)-6-ethyldecahydro-5-hydroxy-4; 6; 9; 10-tetramethyl-1-oxo-3a; 9-propano-3aH-cyclopentacycloocten-8-yl ester; 14-O- (5- (2-Amino1; 3; 4-triazolyl) thioacetyl) dihydromutilin; Antibiotic TDM 85-530] |
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| Gene, Accession, CAS # | CAS: 76530-44-4 |
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| Catalog # | MBS845469 |
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| Price | |
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| Order / More Info | Azamulin from MYBIOSOURCE INC. |
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| Product Specific References | n/a |
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