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| Product Name | Nebivolol hydrochloride |
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| Description | Highly selective β1-adrenoceptor antagonist (Ki values are 0.88, 20, 44, 700, 1160, 2400 and 4000 nM at β1, 5-HT1A, β2, 5-HT2, α1, H1 and D2 receptors respectively). Induces vasodilation via a nitric oxide- and cGMP-dependent mechanism (EC50 = 11.36 μM in renal arteries) and displays antihypertensive activity in vivo. GRK/β -arrestin biased agonist at the β2 adrenoceptor. Purity 98%. MW (observed): 441.9 |
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| Size | 50 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (±)-[2R*(1S*5S*(S*))]-α,α'-[Iminobis(methylene)bis(6-fluoro-3,4-dihydro-2H-1-benzopyran-2-methanol) |
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| Gene, Accession, CAS # | CAS: 152520-56-4 |
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| Catalog # | 3517/50 |
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| Order / More Info | Nebivolol hydrochloride from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 26306764 |
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| 产品资料 |
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