产品详情 |
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Product Name | Tariquidar dihydrochloride |
Description | Potent P-glycoprotein (P-gp) inhibitor (IC50 = 5.1 nM). Reverses drug resistance in multiple MDR cell lines. Acts as a substrate for breast cancer resistance protein (BCRP) at low concentrations and acts as an inhibitor of BCRP when used at >100 nM concentration. Potentiates the cytotoxic effects of doxorubicin (Cat. No. 2252) and mitoxantrone (Cat. No. 4250) in vitro. Purity 98%. MW (observed): 719.66 |
Size | 50 mg |
Concentration | n/a |
Applications | n/a |
Other Names | N-[2-[[[4-[2-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl]phenyl]amino]carbonyl]-4,5-dimethoxyphenyl]-3-quinolinecarbxamide dihydrochloride |
Gene, Accession, CAS # | n/a |
Catalog # | 5757/50 |
Price | |
Order / More Info | Tariquidar dihydrochloride from TOCRIS BIOSCIENCE
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Product Specific References | n/a |
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