| 产品详情 |
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| Product Name | EPZ011989 |
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| Description | MW: 605.82. Purity ≥98% by HPLC. EPZ011989 is a potent EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutated EZH2. It displays 15-fold selectivity for EZH2 over EZH1 and is without effect against an array of other lysine methyltransferases. EPZ011989 demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphoma. |
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| Size | 5 mg, 25 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | [N- ( (4; 6-dimethyl-2-oxo-1; 2-dihydropyridin-3-yl) methyl)-3- (ethyl ( (1r; 4r)-4- ( (2-methoxyethyl) (methyl) amino) cyclohexyl) amino)-2-methyl-5- (3-morpholinoprop-1-yn-1-yl) benzamide] |
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| Gene, Accession, CAS # | CAS: 1598383-40-4 |
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| Catalog # | MBS846363 |
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| Price | |
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| Order / More Info | EPZ011989 from MYBIOSOURCE INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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