产品名称 CTEP - RO 4956371
产品货号 Axon 1972 CAS [871362-31-1] MF C19H13ClF3N3OMW 391.77 Purity: 99% Soluble in DMSO Description Potent, orally bioavailable, long lasting and selective mGluR5 allosteric antagonist or negative allosteric modulator; CTEP binds mGluR5 with low nanomolar affinity and shows >1000-fold selectivity against other targets, including all known mGlu receptorsCTEP has considerably improved properties over older mGluR5 antagonists such as MPEP (Axon 1222) and Fenobam (Axon 1345) KEYWORDS: CTEP | supplier | NAM of mGluR5 | RO 4956371 | RO4956371 | CAS [871362-31-1] | Glutamate | mGluR5 | NAM | allosteric modulator | mpep | fenobam | long lasting
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CTEP - RO 4956371

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1972

CAS [871362-31-1]

MF C19H13ClF3N3O
MW 391.77

  • Purity: 99%
  • Soluble in DMSO

CTEP

Description

Potent, orally bioavailable, long lasting and selective mGluR5 allosteric antagonist or negative allosteric modulator; CTEP binds mGluR5 with low nanomolar affinity and shows >1000-fold selectivity against other targets, including all known mGlu receptorsCTEP has considerably improved properties over older mGluR5 antagonists such as MPEP (Axon 1222) and Fenobam (Axon 1345)

KEYWORDS: CTEP | supplier | NAM of mGluR5 | RO 4956371 | RO4956371 | CAS [871362-31-1] | Glutamate | mGluR5 | NAM | allosteric modulator | mpep | fenobam | long lasting

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