| 产品名称 | BD 1063 dihydrochloride |
| 产品货号 | Axon 2088 CAS [206996-13-6 ] MF C13H18Cl2N2.2HClMW 346.12 Purity: 100% Soluble in water and DMSO Description Potent and selective sigma-1 (σ-1) receptor antagonist (Ki=9 nM); about 50-fold more selective for sigma-1 over sigma-2 and >100-fold more selective over 9 other tested neurotransmitter receptors; shown to antagonize cocaine efffects References Certificates Categories Extra info V Sabino et al. The σ-Receptor Antagonist BD-1063 Decreases Ethanol Intake and Reinforcement in Animal Models of Excessive Drinking. Neuropsychopharmacology 34.6 (2008): 1482-1493. KA McCracken et al. Novel σ receptor ligands attenuate the locomotor stimulatory effects of cocaine. Eur. J. Pharmacol. 1995, 365(1), 35-38. FP Monnet et al. Neurosteroids, via sigma receptors, modulate the [3H] norepinephrine release evoked by N-methyl-D-aspartate in the rat hippocampus. Proc. Nat. Acad. Sci. 1995, 92(9), 3774-3778. Certificate of Analysis Material Safety Data Sheet CNS Sigma Unclassified Selective sigma-1 (σ-1) receptor antagonist Chemical name 1-(3,4-dichlorophenethyl)-4-methylpiperazine dihydrochloride Parent CAS No. [150208-28-9] Order Size Unit Price Stock 10 mg €75.00 In Stock |
| 产品价格 | 现货询价，电话：010-67529703 |
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| 产品品牌 | axonmedchem |
| 产品概述 | |
| 产品详情 |
BD 1063 dihydrochlorideAxon 2088 CAS [206996-13-6 ] MF C13H18Cl2N2.2HCl
Description
Potent and selective sigma-1 (σ-1) receptor antagonist (Ki=9 nM); about 50-fold more selective for sigma-1 over sigma-2 and >100-fold more selective over 9 other tested neurotransmitter receptors; shown to antagonize cocaine efffects
Selective sigma-1 (σ-1) receptor antagonist
Chemical name1-(3,4-dichlorophenethyl)-4-methylpiperazine dihydrochloride Parent CAS No.[150208-28-9] |
| 产品资料 |
