产品名称

SA 4503 - Cutamesine

产品货号

Axon 1767 CAS [165377-44-6] MF C23H32N2O2.2HClMW 441.43 Purity: 99% Soluble in water Description Potent and selective sigma-1 receptor agonist; showing high affinity (IC50=17.4 nM) for sigma-1 and 100 fold less affinity for sigma-2. KEYWORDS: SA 4503 | supplier | Sigma-1 antagonist | Cutamesine | SA4503 | SA-4503 | CAS [165377-44-6] | [165377-43-5] | Sigma Receptor Substrates | Sigma-1 | Antagonist | Receptors

产品价格

现货询价，电话：010-67529703

产品规格

产品品牌

axonmedchem

产品概述

产品详情

SA 4503 - Cutamesine

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 1767

CAS [165377-44-6]

MF C23H32N2O2.2HCl
MW 441.43

Purity: 99%
Soluble in water

SA 4503

Description

Potent and selective sigma-1 receptor agonist; showing high affinity (IC50=17.4 nM) for sigma-1 and 100 fold less affinity for sigma-2.

KEYWORDS: SA 4503 | supplier | Sigma-1 antagonist | Cutamesine | SA4503 | SA-4503 | CAS [165377-44-6] | [165377-43-5] | Sigma Receptor Substrates | Sigma-1 | Antagonist | Receptors

K Matsuno et al. Binding properties of SA4503, a novel and selective sigma 1 receptor agonist. Eur. J. Pharmacol. 1996, 306(1-3), 271–279.

G Skuza and Z Rogóz. The synergistic effect of selective sigma receptor agonists and uncompetitive NMDA receptor antagonists in the forced swim test in rats. J. Physiol. Pharmacol. 2006, 57(2), 217–229.

CNS Sigma Unclassified

Sigma-1 receptor antagonist

Chemical name

1-(3,4-dimethoxyphenethyl)-4-(3-phenylpropyl)piperazine dihydrochloride

Parent CAS No.

[165377-43-5]

产品资料