产品名称

SR 141716 hydrochloride - Rimonabant hydrochloride

产品货号

Axon 1220 CAS [158681-13-1] MF C22H21Cl3N4O.HClMW 500.25 Purity: 99% Soluble in DMSO and Ethanol Description Selective, potent and orally active antagonist of the cannabinoid CB1 receptor with a long duration of action (Ki value 2 nM). KEYWORDS: SR 141716 hydrochloride | supplier | CB1 antagonist | Rimonabant hydrochloride | supplier | SR141716 | CAS [158681-13-1] | [168273-06-1] | Cannabinoids | CB1 | Antagonist | metabolism | gastrointestinal motility | obesity | food intake

产品价格

现货询价，电话：010-67529703

产品规格

产品品牌

axonmedchem

产品概述

产品详情

SR 141716 hydrochloride - Rimonabant hydrochloride

Based on 16 reference(s) in Google Scholar 9 10 16

Axon 1220

CAS [158681-13-1]

MF C22H21Cl3N4O.HCl
MW 500.25

Purity: 99%
Soluble in DMSO and Ethanol

SR 141716 hydrochloride

Description

Selective, potent and orally active antagonist of the cannabinoid CB1 receptor with a long duration of action (Ki value 2 nM).

KEYWORDS: SR 141716 hydrochloride | supplier | CB1 antagonist | Rimonabant hydrochloride | supplier | SR141716 | CAS [158681-13-1] | [168273-06-1] | Cannabinoids | CB1 | Antagonist | metabolism | gastrointestinal motility | obesity | food intake

J Simiand et al. SR 141716, a CB1 cannabinoid receptor antagonist, selectively reduces sweet food intake in marmoset. Behav. Pharmacol. 1998, 9(2), 179-81.

M Rinaldi-Carmona et al. Biochemical and pharmacological characterisation of SR141716A, the first potent and selective brain cannabinoid receptor antagonist. Life Sci. 1995;56(23-24):1941-7.

Cardiovascular CNS Diabetes & Metabolism Pain & Inflammation CB1 A13

CB1 antagonist

Chemical name

5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide hydrochloride

Parent CAS No.

[168273-06-1]

产品资料