| 产品详情 |
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| Product Name | AKR1C3 Inhibitor I |
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| Description | A highly potent and selective inhibitor of the type 5 17-β-hydroxysteroid dehydrogenase AKR1C3. In repeat assays it showed an IC50 of 0.013 ± 0.003 µM for AKR1C3, compared with 20.3 ± 3.8 µM against AKR1C1 and >30 µM against AKR1C2 and AKR1C4. This inhibitor also showed displays potency in a cellular assay, blocking the ability of AKR1C3 to metabolize a proven substrate. Does not display any COX (cyclooxygenase) inhibition at 10 µM in whole blood assay. MW: 317.36. Purity ≥98% by HPLC |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 3-(3,4-Dihydroisoquinolin2(1H)-ylsulfonyl)benzoic acid |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 2403-5 |
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| Price | |
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| Order / More Info | AKR1C3 Inhibitor I from BIOVISION, INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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