| 产品详情 |
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| Product Name | BRD9539 |
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| Description | Purity ≥98%. MW: 399.44. BRD9539 is a specific inhibitor of euchromatin histone methyltransferase G9a (EHMT2). EHMT2 catalyzes the methylation of lysine 9 on histone H3. BRD9539 inhibits EHMT2 with an IC50 of 6.3 µM. It also inhibits methyl transferase PRC2 with a similar IC50. It is the methyl-ester analogue of BRD4770. It is more potent than BRD4770 in enzyme assays but does not show activity in cell-based assays, probably due to impaired cell permeability compared to that of BRD4770. |
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| Size | 1 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | BRD9539; 2-benzamido-1-(3-phenylpropyl)benzimidazole-5-carboxylic acid |
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| Gene, Accession, CAS # | CAS: 1374601-41-8 |
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| Catalog # | B2810-1 |
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| Price | |
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| Order / More Info | BRD9539 from BIOVISION, INC. |
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| Product Specific References | n/a |
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