| 产品详情 |
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| Product Name | EPZ011989 |
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| Description | EPZ011989 is a potent EZH2 inhibitor with Ki values that are less than 3 nM for wild type and Tyr646 mutated EZH2. It displays 15-fold selectivity for EZH2 over EZH1 and is without effect against an array of other lysine methyltransferases. EPZ011989 demonstrates significant tumor growth inhibition in a mouse xenograft model of human B cell lymphoma. MW: 605.82. Purity ≥98% by HPLC |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl((1r,4r)-4-((2-methoxyethyl)(methyl)amino)cyclohexyl)amino)-2-methyl-5-(3-morpholinoprop-1-yn-1-yl)benzamide |
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| Gene, Accession, CAS # | CAS: 1598383-40-4 |
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| Catalog # | B1221-5 |
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| Price | |
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| Order / More Info | EPZ011989 from BIOVISION, INC. |
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| Product Specific References | n/a |
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| 产品资料 |
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