产品详情 |
Edit |   |
Product Name | Methoctramine |
Description | A selective muscarinic M2 receptor antagonist (IC50 = 6.1 nM in CHO-K1 cell membranes); selective for M2 over M1, M3, M4, and M5 receptors (IC50s = 92, 770, 260, and 217 nM, respectively); inhibits acetylcholine-induced reductions in isolated guinea pig tracheal tube contractions in vitro (1 µM); inhibits bradycardia and bronchoconstriction induced by acetylcholine in guinea pigs (ED50s = 38 and 81 nmol/kg, respectively); suppresses oxotremorine M-induced bladder overactivity in a rat model of spinal cord injury |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 104807-40-1 M-2 1 3 4 5 CHOK1 |
Gene, Accession, CAS # | CAS: 104807-46-7 |
Catalog # | 24317-10 |
Price | |
Order / More Info | Methoctramine from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |
产品资料 |
|
|