产品名称 PQ 69 from TOCRIS BIOSCIENCE
产品货号 5351/50
产品价格 现货询价,电话:010-67529703
产品规格 50 mg
产品品牌 TOCRIS BIOSCIENCE
产品概述
产品详情
Edit&nbsp
Product NamePQ 69
DescriptionPotent and selective A1 receptor inverse agonist. Exhibits high binding affinity at A1 receptor (Ki values are 0.07 and 0.96 nM for rat and human receptors respectively). Reduces basal [35S]-GTPγS binding 44.6% (IC50 = 0.19 nM). Antagonizes the effects of A1 agonist R-PIA (IC50 = 18.3 nM) and exhibits competitive antagonism on CCPA -induced tracheal contractions ex vivo. Displays 217- fold selectively over hA2A receptor and >1000-fold selectivity over hA3 receptor. Purity 98%. MW (observed): 350.39
Size50 mg
Concentrationn/a
Applicationsn/a
Other Names4-(Butylamino)-2-(3-fluorophenyl)-1,2-dihydro-3H-pyrazolo[4,3-c]quinolin-3-one
Gene, Accession, CAS #CAS: 910045-32-8
Catalog #5351/50
Price
Order / More InfoPQ 69 from TOCRIS BIOSCIENCE
Product Specific Referencesn/a
产品资料