| 产品详情 |
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| Product Name | Asimadoline |
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| Description | A potent κ-opioid receptor agonist (IC50s = 5.6 and 1.2 nM for guinea pig and human receptors, respectively); is 501- and 498-fold selective for κ-opioid over µ- and δ-opioid receptors, respectively; is spasmolytic in isolated rat duodenum (IC50 = 4.2 µM) and inhibits spontaneous contractions of isolated rat uterus (IC50 = 12.7 µM); reduces joint damage in a rat model of CFA-induced arthritis; reduces the abdominal withdrawal reflex in a model of visceral pain induced by colonic distension in wild-type mice at 25 mg/kg |
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| Size | 1 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | EMD 61753 |
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| Gene, Accession, CAS # | CAS: 153205-46-0 |
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| Catalog # | 26411-1 |
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| Order / More Info | Asimadoline from CAYMAN CHEMICAL COMPANY |
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| Product Specific References | n/a |
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| 产品资料 |
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